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ΤύποςΗμερομηνίαΤίτλοςΔημιουργόςΠλήρες κείμενο
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2008Crystallographic and computational studies on 4-phenyl-N-(beta-D-glucopyranosyl)-1H-1,2, 3-triazole-1-acetamide, an inhibitor of glycogen phosphorylase: Comparison with alpha-D-glucose, N-acetyl-beta-D-glucopyranosylamine and N-benzoyl-N '-beta-D-glucopyranosyl urea bindingAlexacou, Kyra-Melinda; Hayes, Joseph M.; Tiraidis, Costas; Ζωγράφος, Σπύρος Ε.; Λεωνίδας, Δημήτρης Δ.; Χρυσίνα, Ευαγγελία Δ.; Archontis, Georgios; Οικονομάκος, Νίκος Γ.; Paul, Jashuva V.; Varghese, Babu; Loganathan, Duraikkannu
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2008Naturally occurring pentacyclic triterpenes as inhibitors of glycogen phosphorylase: Synthesis, structure-activity relationships, and X-ray crystallographic studiesWen, Xiaoan; Sun, Hongbin; Liu, Jun; Cheng, Keguang; Zhang, Pu; Zhang, Liying; Hao, Jia; Zhang, Luyong; Ni, Peizhou; Ζωγράφος, Σπύρος Ε.; Λεωνίδας, Δημήτρης Δ.; Alexacou, Kyra-Melinda; Gimisis, Thanasis; Hayes, Joseph M.; Οικονομάκος, Νίκος Γ.
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2009Amide-1,2,3-triazole bioisosterism: the glycogen phosphorylase caseΧρυσίνα, Ευαγγελία Δ.; Bokor, Eva; Alexacou, Kyra-Melinda; Charavgi, Maria-Despoina; Oikonomakos, George N.; Ζωγράφος, Σπύρος Ε.; Λεωνίδας, Δημήτρης Δ.; Οικονομάκος, Νίκος Γ.; Laszlo, Somsak
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2009Glucose-based spiro-isoxazolines: A new family of potent glycogen phosphorylase inhibitorsBenltifa, Mahmoud; Hayes, Joseph M.; Vidal, Sebastien; Gueyrard, David; Goekjian, Peter G.; Praly, Jean-Pierre; Kizilis, Gregory; Tiraidis, Costas; Alexacou, Kyra-Melinda; Χρυσίνα, Ευαγγελία Δ.; Ζωγράφος, Σπύρος Ε.; Λεωνίδας, Δημήτρης Δ.; Archontis, Georgios; Οικονομάκος, Νίκος Γ.
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2010Synthesis of new glycosyl biuret and urea derivatives as potential glycoenzyme inhibitorsFelfoldi, Nora; Toth, Marietta; Χρυσίνα, Ευαγγελία Δ.; Charavgi, Maria-Despoina; Alexacou, Kyra-Melinda; Somsak, Laszlo
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2010Glycogen phosphorylase inhibitor identification targeting the inhibitor binding site using virtual screening and experimental validationZhong, Shijun; Alexacou, Kyra-Melinda; Charavgi, Marianna A.; Tiraidis, Costas; Ζωγράφος, Σπύρος Ε.; Λεωνίδας, Δημήτρης Δ.; Χρυσίνα, Ευαγγελία Δ.; Οικονομάκος, Νίκος Γ.; MacKerell, Alexander D., Jr.
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2010The binding of beta-D-glucopyranosyl-thiosemicarbazone derivatives to glycogen phosphorylase: A new class of inhibitorsAlexacou, Kyra-Melinda; Tenchiu (Deleanu), Alia-Cristina; Χρυσίνα, Ευαγγελία Δ.; Charavgi, Maria-Despoina; Κώστας, Ιωάννης Δ.; Ζωγράφος, Σπύρος Ε.; Οικονομάκος, Νίκος Γ.; Λεωνίδας, Δημήτρης Δ.
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2011Halogen-substituted (C-beta-D-glucopyranosyl)-hydroquinone regioisomers: Synthesis, enzymatic evaluation and their binding to glycogen phosphorylaseAlexacou, Kyra-Melinda; Zhang, Yun Zhi; Praly, Jean-Pierre; Ζωγράφος, Σπύρος Ε.; Χρυσίνα, Ευαγγελία Δ.; Οικονομάκος, Νίκος Γ.; Λεωνίδας, Δημήτρης Δ.
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2012N-(4-Substituted-benzoyl)-N '-(beta-D-glucopyranosyl)ureas as inhibitors of glycogen phosphorylase: Synthesis and evaluation by kinetic, crystallographic, and molecular modelling methodsVeronika Nagy; Nora Felfoeldi; Balint Konya; Praly, Jean-Pierre; Tibor Docsa; Pal Gergely; Χρυσίνα, Ευαγγελία Δ.; Tiraidis, Costas; Kosmopoulou, Magda N.; Alexacou, Kyra-Melinda; Konstantakaki, Maria; Λεωνίδας, Δημήτρης Δ.; Ζωγράφος, Σπύρος Ε.; Οικονομάκος, Νίκος Γ.; Kozmon, Stanislav; Tvaroska, Igor; Laszlo Somsak
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